Compile Data Set for Download or QSAR
Found 81 of ic50 data for polymerid = 3971,50000237
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of [3H]-ATRA-Hl60 binding to Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23T9GFVPubMedMMDB
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50075879(4-(2,2-Dimethyl-4-p-tolyl-2H-1-thia-anthracen-6-yl...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Antagonistic activity against RAR gamma in transcriptional activation assay with 3.2 nM TTNPBMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26Q1WFPPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)copy SMILEScopy InChI
Affinity DataIC50: 0.620nMAssay Description:Binding affinity against Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2028QSBPubMedMMDB
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50084832(4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quino...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Binding affinity for Retinoic Acid Receptor gamma (RAR gamma)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50075880(4-(5,5-Dimethyl-8-p-tolyl-5,6-dihydro-anthracen-2-...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Binding affinity of [3H]- RA to baculovirus expressed human Retinoic acid receptor betaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26Q1WFPPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50075877(4-[5,5-Dimethyl-8-(5-methyl-thiophen-2-yl)-5,6-dih...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Antagonistic activity against RAR alpha in transcriptional activation assay with 32 nM TTNPBMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26Q1WFPPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50075878(4-(2,2-Dimethyl-4-p-tolyl-2H-benzo[g]chromen-7-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Binding affinity of [3H]- RA to baculovirus expressed human Retinoic acid receptor betaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26Q1WFPPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50097821(4-{(E)-4-[2-(4-Ethyl-phenyl)-6,6-dimethyl-cyclohex...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Antagonist activity of TTNPB (10 nM) function at retinoic acid receptor betaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2348JN3PubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50029774(4-(5,5-Dimethyl-8-p-tolyl-5,6-dihydro-naphthalen-2...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Binding affinity towards retinoic acid receptor alpha was determined using [3H]-ATRA (5 nM) as radioligandMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2348JN3PubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50084830(4-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quino...)copy SMILEScopy InChI
Affinity DataIC50: 3.60nMAssay Description:Binding affinity for Retinoic Acid Receptor gamma (RAR gamma)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50075876(4-[2,2-Dimethyl-4-(5-methyl-thiophen-2-yl)-2H-benz...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Antagonistic activity against RAR gamma in transcriptional activation assay with 3.2 nM TTNPBMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26Q1WFPPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50084831(4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quino...)copy SMILEScopy InChI
Affinity DataIC50: 4.60nMAssay Description:Binding affinity for Retinoic Acid Receptor gamma (RAR gamma)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50097823(4-[(E)-4-(6,6-Dimethyl-2-p-tolyl-cyclohex-1-enyl)-...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Antagonist activity of TTNPB (10 nM) function at retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2348JN3PubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Binding affinity against retinoic Acid gamma receptor using [3H]- -9-cis-Retinoic Acid in competitive binding assayMore data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50084829(4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quino...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Binding affinity for Retinoic Acid Receptor gamma (RAR gamma)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Binding affinity against retinoic Acid gamma receptor using [3H]- -9-cis-Retinoic Acid in competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20V8BT5PubMedMMDB
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50084833(4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-napht...)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Binding affinity for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50032219((E)-4-(2-(5,5,8,8-tetramethyl-5,6,7,8-tetrahydrona...)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Binding affinity against retinoic Acid gamma receptor using [3H]- -9-cis-Retinoic Acid in competitive binding assayMore data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50084834(4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quino...)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Binding affinity for Retinoic Acid Receptor gamma (RAR gamma)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50097820(4-[(E)-4-(3,3-Dimethyl-6-p-tolyl-cyclohexa-1,5-die...)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Antagonist activity of TTNPB (10 nM) function at retinoic acid receptor alphaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2348JN3PubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50296049((2E,4E)-2,4-dimethyl-5-(6,6,9,9-tetramethyl-4-oxo-...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Displacement of radioligand from RARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58MD3PubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50084837(4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quino...)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Binding affinity for Retinoic Acid Receptor gamma (RAR gamma)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50044099(4-[(E)-2-(3-Ethyl-5,5,8,8-tetramethyl-5,6,7,8-tetr...)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Binding affinity against retinoic Acid gamma receptor using [3H]- -9-cis-Retinoic Acid in competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20V8BT5PubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50084835(4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quino...)copy SMILEScopy InChI
Affinity DataIC50: 310nMAssay Description:Binding affinity for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4P4MPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50097822(4-{(E)-4-[2-(4-tert-Butyl-phenyl)-6,6-dimethyl-cyc...)copy SMILEScopy InChI
Affinity DataIC50: 331nMAssay Description:Antagonist activity of TTNPB (10 nM) function at retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2348JN3PubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50032221(4-[(E)-2-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro...)copy SMILEScopy InChI
Affinity DataIC50: 645nMAssay Description:Binding affinity against retinoic Acid gamma receptor using [3H]- -9-cis-Retinoic Acid in competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20V8BT5PubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203459(CHEMBL3894222)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50044098(4-[(E)-2-(3-Isopropyl-5,5,8,8-tetramethyl-5,6,7,8-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity against retinoic Acid gamma receptor using [3H]- -9-cis-Retinoic Acid in competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20V8BT5PubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203544(CHEMBL3928131)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203542(CHEMBL3218921)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203508(CHEMBL3968165)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203514(CHEMBL3977144)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203516(CHEMBL3967961)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203543(CHEMBL3951385)copy SMILEScopy InChI
Affinity DataIC50: 2.70E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50099474(4-[5-(8-Isopropyl-4-phenyl-quinolin-2-yl)-1H-pyrro...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonistic activity of the compound was evaluated in terms of inhibition of Retinoic acid receptor gamma transactivation by ATRA (50 nM); Not detec...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26M3643PubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203509(CHEMBL3948459)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203504(CHEMBL3938404)copy SMILEScopy InChI
Affinity DataIC50: 3.80E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203490(CHEMBL3905660)copy SMILEScopy InChI
Affinity DataIC50: 4.10E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203539(CHEMBL3950318)copy SMILEScopy InChI
Affinity DataIC50: 4.20E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203518(CHEMBL3942787)copy SMILEScopy InChI
Affinity DataIC50: 4.40E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203499(CHEMBL3947885)copy SMILEScopy InChI
Affinity DataIC50: 4.50E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203517(CHEMBL3933815)copy SMILEScopy InChI
Affinity DataIC50: 5.60E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203503(CHEMBL3982499)copy SMILEScopy InChI
Affinity DataIC50: 5.70E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203515(CHEMBL3920454)copy SMILEScopy InChI
Affinity DataIC50: 6.20E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203460(CHEMBL3956929)copy SMILEScopy InChI
Affinity DataIC50: 6.80E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203488(CHEMBL3957141)copy SMILEScopy InChI
Affinity DataIC50: 6.80E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203462(CHEMBL3931161)copy SMILEScopy InChI
Affinity DataIC50: 7.20E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203513(CHEMBL3913238)copy SMILEScopy InChI
Affinity DataIC50: 7.60E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203502(CHEMBL3940207)copy SMILEScopy InChI
Affinity DataIC50: 7.70E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Eisai Co. Ltd.

Curated by ChEMBL
LigandPNGBDBM50203500(CHEMBL3986751)copy SMILEScopy InChI
Affinity DataIC50: 8.40E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
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